(E/Z)-CLH304a - HY-129636A
Catalog #
HY-129636A
(E/Z)-CLH304a (GABAB receptor antagonist 1) is a mixture of (E)-CLH304a and (Z)-CLH304a. (E)-CLH304a (CLH304a; HY-129636) is a specific and noncompetitive GABAB receptor negative allosteric modulator (NAM). CLH304a inhibits Baclofen (HY-B0007)-induced ERK1/2 phosphorylation in HEK293 cells overexpressing GABAB receptors[1][2].
| Datasheet URL | http://file.medchemexpress.com/batch_PDF/HY-129636A/E-Z-CLH304a-DataSheet-MedChemExpress.pdf |
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| Quantity | Getquote |
| Shipping | Room temperature |
| Application | Neuroscience-Neuromodulation |
| Alternative Names | GABAB receptor antagonist 1 |
| CAS | 797-17-1 |
| MWT | 304.38 |
| Solubility | DMSO : ≥ 200 mg/mL |
| Clinical Information | No Development Reported |
| Target | ERK;GABA Receptor |
| Application: | Neuroscience-Neuromodulation |
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