Antihistamine-1 - HY-100238

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Catalog #
HY-100238
Ab 86,00 €
Antihistamine-1 is a H1-antihistamine (Ki=6.9 nM) with acceptable blood-brain barrier penetration and also an inhibitor of CYP2D6 and hERG channel with IC50s of 5.4 and 0.8 μM, respectively.
Weitere Informationen
Datasheet URL http://file.medchemexpress.com/batch_PDF/HY-100238/Antihistamine-1-DataSheet-MedChemExpress.pdf
Shipping Room Temperature
Application Metabolism-sugar/lipid metabolism
CAS 1186430-60-3
Storage -20°C, 3 years; 4°C, 2 years (Powder)
MWT 389.47
Solubility DMSO : 25 mg/mL (ultrasonic;warming;heat to 60°C)
Clinical Information No Development Reported
Target Cytochrome P450;Histamine Receptor;Potassium Channel
Applications
Application: Metabolism-sugar/lipid metabolism

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