I-BET762 carboxylic acid - HY-107443

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Catalog #
HY-107443
Ab 83,00 €
I-BET762 carboxylic acid (Molibresib carboxylic acid) is an I-BET762-based warhead ligand for conjugation reactions of PROTAC targeting on BET. I-BET762 carboxylic acid (Molibresib carboxylic acid) is a BRD4 inhibitor with a pIC50 of 5.1[1].
Weitere Informationen
Datasheet URL http://file.medchemexpress.com/batch_PDF/HY-107443/I-BET762-carboxylic-acid-DataSheet-MedChemExpress.pdf
Shipping Room Temperature
Application Cancer-programmed cell death
Alternative Names Molibresib carboxylic acid; GSK525762A carboxylic acid; PROTAC BRD4-binding moiety 2
CAS 1300019-38-8
Storage -20°C, 3 years; 4°C, 2 years (Powder)
MWT 396.83
Solubility DMSO : 200 mg/mL (ultrasonic)
Clinical Information No Development Reported
Target Epigenetic Reader Domain;Ligands for Target Protein for PROTAC
Applications
Application: Cancer-programmed cell death

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