PROTAC ERα Degrader-2 - HY-111846

Nur noch %1 verfügbar
Catalog #
HY-111846
Ab 527,00 €
PROTAC ERα Degrader-2 comprises a IAP ligand binding group, a linker and an estrogen receptor α (ERα) binding group. PROTAC ERα Degrader-2 is an ERα degrader. Maximal ERα degradation at 30 μM concentration in human mammary tumor MCF7 cells. Degradation inducers based on cIAP1 are called specific and non-genetic IAP-dependent protein erasers (SNIPERs)[1].
Weitere Informationen
Datasheet URL http://file.medchemexpress.com/batch_PDF/HY-111846/PROTAC-ERα-Degrader-2-DataSheet-MedChemExpress.pdf
Shipping Blue Ice
Application Cancer-programmed cell death
CAS 1351169-29-3
Storage -20°C (Powder, stored under nitrogen)
MWT 763.96
Solubility DMSO : 200 mg/mL (ultrasonic)
Clinical Information No Development Reported
Target Estrogen Receptor/ERR;PROTACs;SNIPERs
Applications
Application: Cancer-programmed cell death

Newsletter
abonnieren

15% Rabatt

erhalten