Casein Kinase inhibitor A86 - HY-123955

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Catalog #
HY-123955
Ab 289,00 €
Casein Kinase inhibitor A86 is a potent and orally active casein kinase 1α (CK1α) inhibitor. Casein Kinase inhibitor A86 also inhibits of CDK7 (TFIIH) and CDK9 (P-TEFb). Casein Kinase inhibitor A861 induces leukemia cell apoptosis, and has potent anti-leukemic activities[1].
Weitere Informationen
Datasheet URL http://file.medchemexpress.com/batch_PDF/HY-123955/Casein-Kinase-inhibitor-A86-DataSheet-MedChemExpress.pdf
Shipping Room Temperature
Application Cancer-Kinase/protease
CAS 2079069-01-3
Storage -20°C, 3 years; 4°C, 2 years (Powder)
MWT 344.43
Solubility DMSO : 12.5 mg/mL (ultrasonic;warming;heat to 60°C)
Clinical Information No Development Reported
Target Apoptosis;Casein Kinase;CDK
Applications
Application: Cancer-Kinase/protease

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