PROTAC CDK2/9 Degrader-1 - HY-130709
Nur noch %1 verfügbar
Catalog #
HY-130709
Ab
775,00 €
PROTAC CDK2/9 Degrader-1 (Compound F3) is a potent dual degrader for CDK2 (DC50=62 nM) and CDK9 (DC50=33 nM). PROTAC CDK2/9 Degrader-1 suppresses prostate cancer PC-3 cell proliferation (IC50=0.12 µM) by effectively blocking the cell cycle in S and G2/M phases. PROTAC CDK2/9 Degrader-1 is a PROTAC by tethering CDK inhibitor with Cereblon ligand[1].
| Datasheet URL | http://file.medchemexpress.com/batch_PDF/HY-130709/PROTAC-CDK2-9-Degrader-1-DataSheet-MedChemExpress.pdf |
|---|---|
| Shipping | Room Temperature |
| Application | Cancer-Kinase/protease |
| CAS | 2408641-24-5 |
| Storage | -20°C, 3 years; 4°C, 2 years (Powder) |
| MWT | 815.84 |
| Solubility | DMSO : 50 mg/mL (ultrasonic) |
| Clinical Information | No Development Reported |
| Target | CDK;PROTACs |
| Application: | Cancer-Kinase/protease |
|---|