Epitinib (succinate) - HY-139300A

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Catalog #
HY-139300A
Ab 300,00 €
Epitinib succinate is an orally active and selective epidermal growth factor receptor tyrosine kinase inhibitor (EGFR-TKI) designed for optimal brain penetration. Epitinib succinate can be used for the research of cancer[1][2]. Epitinib (succinate) is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
Weitere Informationen
Datasheet URL http://file.medchemexpress.com/batch_PDF/HY-139300A/Epitinib-succinate-DataSheet-MedChemExpress.pdf
Shipping Room Temperature
Application Cancer-Kinase/protease
Alternative Names HMPL-813 (succinate)
CAS 2252334-12-4
Storage 4°C (Powder, sealed storage, away from moisture)
MWT 548.59
Solubility DMSO : 12.5 mg/mL (ultrasonic;warming;heat to 60°C)|H2O : < 0.1 mg/mL (ultrasonic;warming;heat to 60°C)
Clinical Information Phase 1
Target EGFR
Applications
Application: Cancer-Kinase/protease

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