PPARγ phosphorylation inhibitor 1 - HY-147705
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Catalog #
HY-147705
Ab
434,00 €
PPARγ phosphorylation inhibitor 1 (Compound 10) is a potent PPARγ binder with the IC50 of 24 nM. PPARγ phosphorylation inhibitor 1 inhibits CDK5-mediated phosphorylation of PPARγ Ser273 with the IC50 of 160 nM. PPARγ phosphorylation inhibitor 1 displays negligible PPARγ agonism in a reporter gene assay. Antidiabetic effects[1].
| Datasheet URL | http://file.medchemexpress.com/batch_PDF/HY-147705/PPARγ-phosphorylation-inhibitor-1-DataSheet-MedChemExpress.pdf |
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| Shipping | Room Temperature |
| Application | Metabolism-protein/nucleotide metabolism |
| CAS | 2882975-84-8 |
| Storage | -20°C, 3 years; 4°C, 2 years (Powder) |
| MWT | 441.26 |
| Solubility | DMSO : 100 mg/mL (ultrasonic;warming;heat to 60°C) |
| Clinical Information | No Development Reported |
| Target | PPAR |
| Application: | Metabolism-protein/nucleotide metabolism |
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