Desfesoterodine - HY-76569
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Catalog #
HY-76569
Ab
186,00 €
Desfesoterodine (PNU-200577) is a potent and selective muscarinic receptor (mAChR) antagonist with a KB and a pA2 of 0.84 nM and 9.14, respectively[1]. Desfesoterodine is a major pharmacologically active metabolite of Tolterodine (PNU-200583; HY-A0024) and Fesoterodine (HY-70053)[2][3]. Desfesoterodine improves cerebral infarction induced detrusor overactivity in rats[4].
| Datasheet URL | http://file.medchemexpress.com/batch_PDF/HY-76569/Desfesoterodine-DataSheet-MedChemExpress.pdf |
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| Shipping | Room Temperature |
| Application | Neuroscience-Neuromodulation |
| Alternative Names | PNU-200577; 5-Hydroxymethyl Tolterodine |
| CAS | 207679-81-0 |
| Storage | -20°C, 3 years; 4°C, 2 years (Powder) |
| MWT | 341.50 |
| Solubility | DMSO : 50 mg/mL (ultrasonic)|H2O : 100 mg/mL (ultrasonic) |
| Clinical Information | Launched |
| Target | mAChR |
| Application: | Neuroscience-Neuromodulation |
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