Bicuculline - HY-N0219
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Catalog #
HY-N0219
Ab
80,00 €
Bicuculline ((+)-Bicuculline) is A competing neurotransmitter GABAA receptor antagonist (IC50=2 μM). Bicuculline also blocks Ca2+ activating potassium (SK) channels and subsequently blocks slow post-hyperpolarization (slow AHP). Bicuculline has anticonvulsant activity. Bicuculline can be used to induce seizures in mice[1][2][3][4].
| Datasheet URL | http://file.medchemexpress.com/batch_PDF/HY-N0219/Bicuculline-DataSheet-MedChemExpress.pdf |
|---|---|
| Shipping | Room Temperature |
| Alternative Names | (+)-Bicuculline |
| CAS | 485-49-4 |
| Storage | 4°C (Powder, protect from light) |
| MWT | 367.35 |
| Solubility | DMSO : 50 mg/mL (ultrasonic)|H2O : < 0.1 mg/mL |
| Clinical Information | No Development Reported |
| Target | GABA Receptor |