EPI-7170 - HY-150102

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Catalog #
HY-150102
Ab 289,00 €
EPI-7170, a ralaniten analogue, is a potent androgen receptor N-terminal structural domain antagonist that blocks the transcriptional activity of full-length AR (FL-AR) and AR splice variants (AR-Vs). EPI-7170 has antitumor effects against enzalutamide resistant castration-resistant prostate cancer (CRPC)[1].
Weitere Informationen
Datasheet URL http://file.medchemexpress.com/batch_PDF/HY-150102/EPI-7170-DataSheet-MedChemExpress.pdf
Shipping Room Temperature
Application Cancer-programmed cell death
CAS 2139288-26-7
Storage 4°C (Powder, sealed storage, away from moisture)
MWT 540.88
Solubility DMSO : 100 mg/mL (ultrasonic)
Clinical Information No Development Reported
Target Androgen Receptor
Applications
Application: Cancer-programmed cell death

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